百灵威五元多杂环砌块 | 咪唑·噻唑·吡唑·三唑等系列全覆盖
2026-07-14 · 推荐产品 · 百灵威授权转载
咪唑、噻唑、吡唑、三唑等含多个杂原子的五元杂环，是药物分子中最常见的核心骨架之一——从抗真菌药（咪唑类）到抗生素（噻唑类），从抗肿瘤药（吡唑类）到抗病毒药（三唑类），其结构多样性和生物活性为药物发现提供了广阔的空间。此外，四唑、噁唑、噁唑烷酮、噻二唑、噁二唑、二噻烷等品种，在药物化学、材料科学和配位化学中同样各具独特应用场景。
从经典的五元杂环偶联到C-H官能团化，这些砌块为药物化学与材料科学提供了丰富的结构起点。
百灵威提供上述五元多杂环砌块，纯度≥95%，稳定供应护航每一步转化。配套常用溶剂与耗材，即用即选，助您高效推进合成路线。
咪唑砌块
| 品名 | CAS | 货号 |
|---|---|---|
| 3-Methyl(triazenyl)imidazole-4-carboxamide, 98% 3-甲基(三氮杂烯基)咪唑-4 甲酰胺 | 3413-72-7 | 618199 |
| 2-Methylimidazole, 99% 2-甲基咪唑 | 693-98-1 | 159278 |
| 1H-Imidazole-2-carboxylic acid, 98% 1H-咪唑-2-羧酸 | 16042-25-4 | 116107 |
| N-Isopropylimidazole, 98% N-异丙基咪唑 | 4532-96-1 | 119534 |
| Tinidazole, 98% 替硝唑 | 19387-91-8 | 153096新 |
| Ethyl 4-(2-Hydroxy-2-propyl)-2-propyl-1H-imidazole-5-carboxylate, 96% 4-(1-羟基-1-甲基乙基)-2-丙基-1H-咪唑-5-羧酸乙酯 | 144689-93-0 | 165648 |
| 1-Ethyl-2-methylimidazole, 98% 1-乙基-2-甲基咪唑 | 21202-52-8 | 1789262 |
| 1-Butyl-2-methylimidazole, 98% 1-丁基-2-甲基咪唑 | 13435-22-8 | 1789263 |
| 1-Ethyl-3-methylimidazolium trifluoroacetate, 98% 1-乙基-3-甲基咪唑三氟乙酸盐 | 174899-65-1 | 187780新 |
| Di(1H-imidazol-1-yl)methane, 97% 二(1H-咪唑-1-基)甲烷 | 84661-56-3 | 1894844 |
| 1,3-Dimethylimidazolium chloride, 98% 1,3-二甲基咪唑氯盐 | 79917-88-7 | 328831 |
噻唑砌块
| 品名 | CAS | 货号 |
|---|---|---|
| 2,4-Dibromothiazole-5-methanol, 97% 2,4-二溴噻唑-5-甲醇 | 170232-68-5 | 1426567 |
| Ethyl benzo[d]thiazole-5-carboxylate, 97% 苯并[d]噻唑-5-甲酸乙酯 | 103261-70-7 | 1515438 |
| 2-(2-Formamidothiazol-4-yl)acetic acid, 97% 2-(2-甲酰氨基噻唑-4-基)乙酸 | 75890-68-5 | 301660 |
| Thiazole-5-carboxaldehyde, 98% 5-噻唑甲醛 | 1003-32-3 | 517926 |
| 2,4-Dichloro-5-cyanothiazole, 97% 2,4-二氯-5-氰基噻唑 | 82554-18-5 | 830973 |
吡唑砌块
| 品名 | CAS | 货号 |
|---|---|---|
| 5-Amino-1-phenylpyrazole, 98% 5-氨基-1-苯基吡唑 | 826-85-7 | 924705 |
| Sacubitril calcium, 98% 沙卡布曲 钙盐 | 1369773-39-6 | 997228 |
| 5-Amino-1-ethylpyrazol, 98% 5-氨基-1-乙基吡唑 | 3528-58-3 | 493314 |
| 1-(2-Methoxyethyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole, 98% 1-(2-甲氧基乙基)-4-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-1H-吡唑 | 847818-71-7 | 1426964 |
| tert-Butyl 3,5-dimethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-carboxylate, 98% 3,5-二甲基-4-(4,4,5,5-四甲基-1,3,2-二氧硼杂环戊烷-2-基)-1H-吡唑-1-羧酸叔丁酯 | 1073354-70-7 | 789336 |
三唑砌块
| 品名 | CAS | 货号 |
|---|---|---|
| 1H-1,2,3-Triazole, 98% 1H-1,2,3-三氮唑 | 288-36-8 | 135039 |
| 3,5-Dibromo-1H-1,2,4-triazole, 99% 3,5-二溴-1H-1,2,4-三唑 | 7411-23-6 | 120698新 |
| 2,6-Dibromo-[1,2,4]triazolo[1,5-a]pyridine, 97% 2,6-溴-[1,2,4]噻唑并[1,5-a]吡啶 | 1401624-81-4 | 1877544 |
| 1,4-Di(4H-1,2,4-triazol-4-yl)benzene, 97% 1,4-二(4H-1,2,4-三唑-4-基)苯 | 681004-60-4 | 2328039 |
| 1-(p-Toluenesulfonyl)-1,2,4-triazole, 98% 1-对甲苯磺酰基-1,2,4-三唑 | 13578-51-3 | 516760 |
| Paclobutrazol, 98% 多效唑 | 76738-62-0 | 122321 |
其他五元多杂环砌块
| 品名 | CAS | 货号 |
|---|---|---|
| 2-Methyl-5-aminotetrazole, 98% 2-甲基-5-氨基四氮唑 | 1553-84-0 | 1355936 |
| 1-Methyl-5-aminotetrazole, 98% 1-甲基-5-氨基四氮唑 | 5422-44-6 | 139439 |
| Pyridino-tetrazole, 98% 吡啶并四氮唑 | 274-87-3 | 2323129 |
| 1,4-Bis(5-phenyl-2-oxazolyl)benzene, 98% 1,4-双(5-苯基-2-恶唑基)苯 | 1806-34-4 | 110604 |
| 5-Ethoxy-4-methyloxazole, 98% 5-乙氧基-4-甲基噁唑 | 5006-20-2 | 147828 |
| (4S,4'S)-2,2'-(Cyclopentane-1,1-diyl)-bis(4-isopropyl-4,5-dihydrooxazole), 95% (4S,4'S)-2,2'-(环戊烷-1,1-二基)-双(4-异丙基-4,5-二氢噁唑) | 1379452-52-4 | 1561126 |
| PNU-120596, 98% PNU-120596, α7 nAChR 阳性变构调节剂 | 501925-31-1 | 1239134 |
| 2-(Bromomethyl)benzo[d]oxazole, 96% 2-溴甲基苯并恶唑 | 73101-74-3 | 1416914 |
| 2-(4-Aminophenyl)benzo[d]oxazol-5-amine, 98% 2-(4-氨基苯基)苯并恶唑-5-胺 | 13676-47-6 | 501559 |
| 4,7-Bis(4-bromophenyl)benzo[c][1,2,5]thiadiazole , 98% 4,7-双(4-溴苯基)苯并[c][1,2,5]噻二唑 | 287966-64-7 | 9380243 |
| 3-(5-Chloro-2-hydroxybenzyl)-5-(4-(trifluoromethyl)-phenyl)-1,3,4-oxadiazol-2(3H)-one, 98% 3-(5-氯-2-羟基苄基)-5-(4-三氟甲基苯基)-1，3，4-二噁唑-2-酮 | 202821-81-6 | 1513107 |
| 2-Phenyl-1,3-dithiane, 98% 2-苯基-1,3-二噻烷 | 5425-44-5 | 958194 |
合成溶剂
| 品名 | CAS | 货号 |
|---|---|---|
| 1,1,1,2-Tetrachloroethane, 98% 1,1,1,2-四氯乙烷 | 630-20-6 | 916866 |
| Triethylamine, 99%, SuperDry, with molecular sieves, Water≤50 ppm, J&Kseal 三乙胺 | 121-44-8 | 919695新 危化品 |
| Dimethyl sulfoxide, 99.5%, AR 二甲基亚砜 | 67-68-5 | 965055 |
| Ethyl acetate, 99.9%, SuperDry, with molecular sieves, Water≤50 ppm, J&KSeal 乙酸乙酯 | 141-78-6 | 920352促 危化品 |
| Acetonitrile, 99.9%, SuperDry, with molecular sieves, water≤50 ppm, J&KSeal 乙腈 | 75-05-8 | 939631促 危化品 |
| 1,2-Dichloroethane, 99.8%, SuperDry, water≤50 ppm, J&Kseal 1,2-二氯乙烷 | 107-06-2 | 981955 危化品 |
| Dichloromethane, 99.9%, SuperDry, with molecular sieves, water≤30 ppm, J&KSeal 二氯甲烷 | 75-09-2 | 908525促 危化品 |
| Tetrahydrofuran, 99.5%, SuperDry, with molecular sieves, stabilized with 250 ppm BHT, Water≤50 ppm, J&KSeal 四氢呋喃 | 109-99-9 | 974643促 危化品 |
耗材
| 品名 | CAS | 货号 |
|---|---|---|
| Magnetic stir bar, PTFE-coated, egg-shaped, A200(8-9mm*20mm), 5 pcs/pack 聚四氟乙烯磁力搅拌子,椭圆型 | / | 978702 |
| 100% Cotton laboratory coats, men, L (170-175cm, 60-70 kg), long-sleeved 纯棉实验服 | / | 992821 |
| Centrifuge tube, 50 mL, vertical, with scale, conical bottom, sterile, 25 pcs/bag, 2 bags/case 离心管 | / | 958546 |
| TLC silica gel plate(fluorescent indicator), HPTLC, GF254, layer thickness 0.2 - 0.25 mm, 75*25 mm, 400 pcs/pack, binder polyacrylate-Na 薄层色谱硅胶板(含荧光) | / | 936755 |
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